Duplessis Martin

Constellation Pharmaceuticals

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论文共 38 篇作者统计合作学者相似作者

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GNE-064: A Potent, Selective, and Orally Bioavailable Chemical Probe for the Bromodomains of SMARCA2 and SMARCA4 and the Fifth Bromodomain of PBRM1

Alexander M. Taylor, Chris Bailey, Lisa D. Belmont,Robert Campbell,Nico Cantone,Alexandre Cote,Terry D. Crawford,Richard Cummings,Kevin DeMent,Martin Duplessis,Megan Flynn,Andrew C. Good,Hon-Ren Huang,Shivangi Joshi,Yves Leblanc,Jeremy Murray,Christopher G. Nasveschuk,Adrianne Neiss,Florence Poy,F. Anthony Romero,Peter Sandy,Yong Tang,Vickie Tsui,Laura Zawadzke,Robert J. Sims,James E. Audia,Steven F. Bellon,Steven R. Magnuson,Brian K. Albrecht,Andrea G. Cochran

Journal of Medicinal Chemistry（2022）

引用4浏览0WOS引用

Design and Synthesis of Styrenylcyclopropylamine LSD1 Inhibitors

Victor S. Gehling,John P. Mcgrath,Martin Duplessis,Avinash Khanna,Francois Brucelle,Rishi G. Vaswani,Alexandre Cote,Jacob Stuckey,Venita Watson,Richard T. Cummings,Srividya Balasubramanian,Priya Iyer, Priyanka Sawant,Andrew C. Good,Brian K. Albrecht,Jean-Christophe Harmange,James E. Audia,Steven F. Bellon,Patrick Trojer,Julian R. Levell

ACS Medicinal Chemistry Letters（2020）

引用17浏览0WOS引用

GNE-371, a Potent and Selective Chemical Probe for the Second Bromodomains of Human Transcription-Initiation-Factor TFIID Subunit 1 and Transcription-Initiation-Factor TFIID Subunit 1-Like

Shumei Wang,Vickie Tsui,Terry D. Crawford,James E. Audia,Daniel Burdick,Maureen H. Beresini,Alexandre Cote,Richard Cummings,Martin Duylessis,E. Megan Flynn,Michael C. Hewitt,Hon-Ren Huang,Hariharan Jayaram,Ying Jiang,Shivangi Joshi,Jeremy Murray,Christopher G. Nasveschuk,Eneida Pardo,Florence Poy,F. Anthony Romero,Yong Tang,Alexander M. Taylor,Jian Wang,Zhaowu Xu,Laura E. Zawadzke,Xiaoyu Zhu,Brian K. Albrecht,Steven R. Magnuson,Steve Bellon,Andrea G. Cochran

Journal of Medicinal Chemistry（2018）

引用11浏览0WOS引用

GNE-886: A Potent and Selective Inhibitor of the Cat Eye Syndrome Chromosome Region Candidate 2 Bromodomain (CECR2)

Terry D Crawford,James E Audia,Steve Bellon,Daniel J Burdick,Archana Bommi-Reddy,Alexandre Côté,Richard T Cummings,Martin Duplessis,E Megan Flynn,Michael Hewitt,Hon-Ren Huang,Hariharan Jayaram,Ying Jiang,Shivangi Joshi,James R Kiefer,Jeremy Murray,Christopher G Nasveschuk, Arianne Neiss,Eneida Pardo,F Anthony Romero,Peter Sandy,Robert J Sims,Yong Tang,Alexander M Taylor,Vickie Tsui,Jian Wang,Shumei Wang,Yongyun Wang,Zhaowu Xu,Laura Zawadzke,Xiaoqin Zhu,Brian K Albrecht,Steven R Magnuson,Andrea G Cochran

ACS medicinal chemistry letters（2017）

引用19浏览0WOS引用

Inhibition of bromodomain-containing protein 9 for the prevention of epigenetically-defined drug resistance

Terry D Crawford,Steffan Vartanian,Alexandre Côté,Steve Bellon,Martin Duplessis,E Megan Flynn,Michael Hewitt,Hon-Ren Huang,James R Kiefer,Jeremy Murray,Christopher G Nasveschuk,Eneida Pardo,F Anthony Romero,Peter Sandy,Yong Tang,Alexander M Taylor,Vickie Tsui,Jian Wang,Shumei Wang,Laura Zawadzke,Brian K Albrecht,Steven R Magnuson,Andrea G Cochran,David Stokoe

Bioorganic & Medicinal Chemistry Letters（2017）

引用29浏览0WOS引用

Discovery of Potent, Orally Bioavailable Inhibitors of Human Cytomegalovirus

Lee Fader,Martine Brault, Jessica Desjardins,Nathalie Dansereau,Louie Lamorte,Sonia Tremblay,Francois Bilodeau,Josee Bordeleau,Martin Duplessis,Vida Gorys,James Gillard, James L. Gleason,Clint James,Marc-Andre Joly,Cyrille Kuhn,Montse Llinas-Brunet,Laibin Luo,Louis Morency,Sebastien Morin,Mathieu Parisien,Maude Poirier,Carl Thibeault,Thao Trinh,Claudio Sturino,Sanjay Srivastava,Christiane Yoakim,Michael Franti

ACS Medicinal Chemistry Letters（2016）

引用4浏览0WOS引用

Diving into the Water: Inducible Binding Conformations for BRD4, TAF1(2), BRD9, and CECR2 Bromodomains

Terry D Crawford,Vickie Tsui,E Megan Flynn,Shumei Wang,Alexander M Taylor,Alexandre Côté,James E Audia,Maureen H Beresini,Daniel J Burdick,Richard Cummings,Les A Dakin,Martin Duplessis,Andrew C Good,Michael C Hewitt,Hon-Ren Huang,Hariharan Jayaram,James R Kiefer,Ying Jiang,Jeremy Murray,Christopher G Nasveschuk,Eneida Pardo,Florence Poy,F Anthony Romero,Yong Tang,Jian Wang,Zhaowu Xu,Laura E Zawadzke,Xiaoyu Zhu,Brian K Albrecht,Steven R Magnuson,Steve Bellon,Andrea G Cochran

JOURNAL OF MEDICINAL CHEMISTRY（2016）

引用87浏览0WOS引用

Identification of (R)-N-((4-methoxy-6-methyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-2-methy L-1-(1-(1-(2,2,2-Trifluoroethyl)Piperidin-4-Yl)Ethyl)-1h-Indole-3-Carbox Amide (Cpi-1205), A Potent and Selective Inhibitor of Histone Methyltransferase Ezh2, Suitable for Phase I Clinical Trials for B-Cell Lymphomas

Rishi G. Vaswani,Victor S. Gehling,Les A. Dakin,Andrew S. Cook,Christopher G. Nasveschuk,Martin Duplessis,Priyadarshini Iyer,Srividya Balasubramanian, Feng Zhao,Andrew C. Good,Robert Campbell,Christina Lee,Nico Cantone,Richard T. Cummings,Emmanuel Normant,Steven F. Bellon,Brian K. Albrecht,Jean-Christophe Harmange,Patrick Trojer,James E. Audia, Ying Zhang,Neil Justin,Shuyang Chen,Jon R. Wilson,Steven J. Gamblin

JOURNAL OF MEDICINAL CHEMISTRYno. 21 (2016): 9928-9941

引用0浏览0引用

Identification of (R)-N-((4-Methoxy-6-methyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-2-methyl-1-(1-(1-(2,2,2-trifluoroethyl)piperidin-4-yl)ethyl)-1H-indole-3-carboxamide (CPI-1205), a Potent and Selective Inhibitor of Histone Methyltransferase EZH2, Suitable for Phase I Clinical Trials for B-Cell Lymphomas

Rishi G Vaswani,Victor S Gehling,Les A Dakin,Andrew S Cook,Christopher G Nasveschuk,Martin Duplessis,Priyadarshini Iyer,Srividya Balasubramanian,Feng Zhao,Andrew C Good,Robert Campbell,Christina Lee,Nico Cantone,Richard T Cummings,Emmanuel Normant,Steven F Bellon,Brian K Albrecht,Jean-Christophe Harmange,Patrick Trojer,James E Audia,Ying Zhang,Neil Justin,Shuyang Chen,Jon R Wilson,Steven J Gamblin

JOURNAL OF MEDICINAL CHEMISTRY（2016）

引用176浏览0WOS引用

176

MODULATORS OF METHYL MODIFYING ENZYMES, COMPOSITIONS AND USES THEREOF

Brian K Albrecht,James E Audia,Andrew S Cook,Les A Dakin,Martin Duplessis,Victor S Gehling,Jeanchristophe Harmange,Christopher G Nasveschuk,Rishi G Vaswani

mag（2015）

引用26浏览0引用

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作者统计

#Papers: 38

#Citation: 956

H-Index: 17

G-Index: 29

Sociability: 5

Diversity: 2

Activity: 3

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