György Miklós Keserű

基本信息

Career Trajectory

Bio

He played a significant role in the development of physicochemical profiling in drug discovery, the concept of compound quality and the improvement of optimization strategies in medicinal chemistry. His results has been acknowledged by the George A Olah Award and the Prous Institute Overton and Meyer Award of the European Federation of Medicinal Chemistry. In 2016 he has been elected as a Fellow (FRSC) of the Royal Society of Chemistry.

Research Interests

Papers共 235 篇Author StatisticsCo-AuthorSimilar Experts

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Contribution of Noncovalent Recognition and Reactivity to the Optimization of Covalent Inhibitors: A Case Study on KRasG12C

Nikolett Peczka,Ivan Randelovic,Zoltan Orgovan,Noemi Csorba,Attila Egyed,Laszlo Petri,Peter Abranyi-Balogh,Marton Gadanecz,Andras Perczel,Jozsef Tovari,Gitta Schlosser,Tamas Takacs,Levente M. Mihalovits,Gyorgy G. Ferenczy,Laszlo Buday,Gyorgy M. Keseru

ACS CHEMICAL BIOLOGYno. 8 (2024): 1743-1756

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Site-Selective Antibody Conjugation with Dibromopyrazines

Denes Szepesi Kovacs, Bettina Pasztor,Peter Abranyi-Balogh,Laszlo Petri,Timea Imre, Jozsef Simon,Eniko Tatrai,Gyorgy Varady,Jozsef Tovari,Peter A. Szijj,Gyorgy M. Keseru

BIOCONJUGATE CHEMISTRYno. 9 (2024): 1373-1379

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Comparative Study of Allosteric GPCR Binding Sites and Their Ligandability Potential

Sonja Peter,Lydia Siragusa, Morgan Thomas, Tommaso Palomba,Simon Cross,Noel M. O'Boyle,David Bajusz,Gyorgy G. Ferenczy,Gyorgy M. Keseru, Giovanni Bottegoni, Brian Bender,Ijen Chen, Chris De Graaf

J Chem Inf Modelno. 21 (2024): 8176-8192

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Molecular Mechanism of Labelling Functional Cysteines by Heterocyclic Thiones

Levente M. Mihalovits,Levente Kollar,David Bajusz,Damijan Knez,Kristof Bozovicar,Timea Imre,Gyorgy G. Ferenczy,Stanislav Gobec,Gyorgy M. Keseru

CHEMPHYSCHEM（2024）

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Mapping Protein Binding Sites by Photoreactive Fragment Pharmacophores

COMMUNICATIONS CHEMISTRYno. 1 (2024)

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Boronic Acid Inhibitors of Penicillin-Binding Protein 1b: Serine and Lysine Labelling Agents

Levente Kollar,Katarina Grabrijan,Martina Hrast Rambaher,Kristof Bozovicar,Timea Imre,Gyorgy G. Ferenczy,Stanislav Gobec,Gyorgy M. Keseru

JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRYno. 1 (2024)

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Novel-Type GABAB PAMs: Structure-Activity Relationship in Light of the Protein Structure

Balazs Kramos,Zsuzsa Hadady,Attila Mako,Gabor Szanto,Nora Felfoldi,Ildiko Magdo,Amrita Agnes Bobok,Imre Bata,Viktor Roman,Andras Visegrady,Gyorgy M. Keseru,Istvan Greiner,Janos Eles

ACS Medicinal Chemistry Letters（2024）

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Exploring Chemical Spaces in the Billion Range: is Docking a Computational Alternative to DNA-Encoded Libraries

Levente M. Mihalovits, Tibor V. Szalai,David Bajusz,Gyorgy M. Keseru

JOURNAL OF CHEMICAL INFORMATION AND MODELING（2024）

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GPCRdb in 2023: State-Specific Structure Models Using AlphaFold2 and New Ligand Resources

Gaspar Pandy-Szekeres,Jimmy Caroli,Alibek Mamyrbekov,Ali A. Kermani,Gyorgy M. Keseru,Albert J. Kooistra,David E. Gloriam

NUCLEIC ACIDS RESEARCH（2023）

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Principal investigator

Papers共 235 篇Author StatisticsCo-AuthorSimilar Experts