Carolyn A. Weigelt

Molecular Structure and Design Research & Development, Bristol-Myers Squibb Company

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论文共 53 篇作者统计合作学者相似作者

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Substituted Diaryl Ether Compounds As Retinoic Acid-Related Orphan Receptor-Gamma T (Ror Gamma T) Agonists

Zheming Ruan,Peter K Park,Donna Wei,Ashok Purandare,Honghe Wan,Daniel O'Malley,Sylwia Stachura,Heidi Perez,Cullen L Cavallaro,Carolyn A Weigelt,John S Sack,Max Ruzanov,Javed Khan,Murali Gururajan,Jessica J Wong,Yanling Huang,Melissa Yarde,Zhuyin Li,Cliff Chen,Huadong Sun,Virna Borowski,Jenny H Xie,Monique Anthony,Michele Agler,Brian E Fink,Lalgudi S Harikrishnan

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS（2021）

引用3浏览0WOS引用

Azatricyclic Inverse Agonists of RORγt That Demonstrate Efficacy in Models of Rheumatoid Arthritis and Psoriasis

Qingjie Liu,Hai-Yun Xiao,Douglas G. Batt,Zili Xiao,Yeheng Zhu,Michael G. Yang, Ning Li,Shiuhang Yip,Peng Li,Dawn Sun,Dauh-Rurng Wu,Max Ruzanov,John S. Sack,Carolyn A. Weigelt,Jinhong Wang,Sha Li,David J. Shuster,Jenny H. Xie,Yunling Song,Tara Sherry,Mary T. Obermeier,Aberra Fura,Kevin Stefanski,Georgia Cornelius,Silvi Chacko,Purnima Khandelwal,Shailesh Dudhgaonkar,Anjuman Rudra,Jignesh Nagar,Venkata Murali,Arun Govindarajan,Rex Denton,Qihong Zhao,Nicholas A. Meanwell,Robert Borzilleri,T. G. Murali Dhar

ACS Medicinal Chemistry Letters（2021）

引用3浏览0WOS引用

Tricyclic-Carbocyclic RORγt Inverse Agonists-Discovery of BMS-986313

Michael G. Yang,Myra Beaudoin-Bertrand,Zili Xiao,David Marcoux,Carolyn A. Weigelt,Shiuhang Yip,Dauh-Rurng Wu,Max Ruzanov,John S. Sack,Jinhong Wang,Melissa Yarde,Sha Li,David J. Shuster,Jenny H. Xie,Tara Sherry,Mary T. Obermeier,Aberra Fura,Kevin Stefanski,Georgia Cornelius,Purnima Khandelwal,Ananta Karmakar,Mushkin Basha,Venkatesh Babu,Arun Kumar Gupta,Arvind Mathur,Luisa Salter-Cid,Rex Denton,Qihong Zhao,T. G. Murali Dhar

Journal of medicinal chemistry（2021）

引用10浏览0WOS引用

A novel MTA non-competitive PRMT5 inhibitor

Rohit Malik,Peter K. Park,Christopher M. Barbieri,Yuval Blat,Steven Sheriff,Carolyn A. Weigelt,Lisa M. Kopcho,Muge Celiktas,Max Ruzanov,Joseph G. Naglich,Jennifer L. Price,Mary Harner,Kevin M. Omalley,Jingjing Deng,William Schmitz,Guo Li,Zheming Ruan,Lan-ying Qin,Gerald J. Duke,Iyoncy Rodrigo,Mark R. Witmer,David G. Harden,Shilpa Demes,Brian J. Arey,Matt Soars,Brian E. Fink,Ashvinikumar V. Gavai,Gregory D. Vite,Charles F. Voliva

CANCER RESEARCH（2021）

引用3浏览0引用

Abstract 1140: A novel MTA non-competitive PRMT5 inhibitor

Rohit Malik,Peter K. Park,Christopher M. Barbieri,Yuval Blat,Steven Sheriff,Carolyn A. Weigelt,Lisa M. Kopcho,Muge Celiktas,Max Ruzanov,Joseph G. Naglich,Jennifer L. Price,Mary Harner,Kevin M. Omalley,JIngjing Deng,William Schmitz,Guo Li,Zheming Ruan,Lan-ying Qin,Gerald J. Duke,Iyoncy Rodrigo,Mark R. Witmer,David G. Harden,Shilpa Demes,Brian J. Arey,Matt Soars,Brian E. Fink,Ashvinikumar V. Gavai,Gregory D. Vite,Charles F. Voliva

Cancer Research（2021）

引用2浏览0引用

Tricyclic Sulfones As Potent, Selective and Efficacious RORγt Inverse Agonists – Exploring C6 and C8 SAR Using Late-Stage Functionalization

Qing Shi,Zili Xiao,Michael G. Yang,David Marcoux,Robert J. Cherney,Shiuhang Yip,Peng Li,Dauh-Rurng Wu,Carolyn A. Weigelt,John Sack,Javed Khan,Max Ruzanov,Jinhong Wang,Melissa Yarde,Mary Ellen Cvijic,Sha Li,David J. Shuster,Jenny Xie,Tara Sherry,Mary Obermeier,Aberra Fura,Kevin Stefanski,Georgia Cornelius,Silvi Chacko,Yue-Zhong Shu,Purnima Khandelwal,John Hynes,Joseph A. Tino,Luisa Salter-Cid,Rex Denton,Qihong Zhao,T. G. Murali Dhar

Bioorganic & medicinal chemistry letters（2020）

引用5浏览0WOS引用

Novel Tricyclic Pyroglutamide Derivatives As Potent RORγt Inverse Agonists Identified Using a Virtual Screening Approach

Qingjie Liu,Douglas G. Batt,Carolyn A. Weigelt,Shiuhang Yip,Dauh-Rurng Wu,Max Ruzanov,John S. Sack,Jinhong Wang,Melissa Yarde,Sha Li,David J. Shuster,Jenny H. Xie,Tara Sherry,Mary T. Obermeier,Aberra Fura,Kevin Stefanski,Georgia Cornelius,Purnima Khandelwal,Joseph A. Tino,John E. Macor,Luisa Salter-Cid,Rex Denton,Qihong Zhao,T. G. Murali Dhar

ACS medicinal chemistry letters（2020）

引用10浏览0WOS引用

Discovery of 2,6-Difluorobenzyl Ether Series of Phenyl ((R)-3-phenylpyrrolidin-3-yl)sulfones As Surprisingly Potent, Selective and Orally Bioavailable RORγt Inverse Agonists

James J-W Duan,Bin Jiang,Zhonghui Lu,Sylwia Stachura,Carolyn A. Weigelt,John S. Sack,Javed Khan,Max Ruzanov,Dauh-Rurng Wu,Melissa Yarde,Ding-Ren Shen,Qihong Zhao,Luisa M. Salter-Cid,Percy H. Carter,T. G. Murali Dhar

Bioorganic & medicinal chemistry letters（2020）

引用3浏览0WOS引用

Discovery of (3S,4s)-3-methyl-3-(4-fluorophenyl)-4-(4-(1,1,1,3,3,3-hexafluoro-2-hydroxyprop-2-yl)phenyl)pyrrolidines As Novel RORγt Inverse Agonists

Bin Jiang,James J. -W. Duan,Sylwia Stachura,Ananta Karmakar,Hemalatha Hemagiri,Dhanya Kumar Raut,Arun Kumar Gupta,Carolyn A. Weigelt,Javed Khan,John S. Sack,Dauh-Rurng Wu,Melissa Yarde,Ding-Ren Shen,Michael A. Galella,Arvind Mathur,Qihong Zhao,Luisa M. Salter-Cid,Percy H. Carter,T. G. Murali Dhar

Bioorganic & medicinal chemistry letters（2020）

引用10浏览0WOS引用

Discovery of BMS-986251: A Clinically Viable, Potent, and Selective RORγt Inverse Agonist

Robert J. Cherney,Lyndon A. M. Cornelius,Anurag Srivastava,Carolyn A. Weigelt,David Marcoux,James J-W Duan,Qing Shi,Douglas G. Batt,Qingjie Liu,Shiuhang Yip,Dauh-Rurng Wu,Max Ruzanov,John Sack,Javed Khan,Jinhong Wang,Melissa Yarde,Mary Ellen Cvijic,Arvind Mathur,Sha Li,David Shuster,Purnima Khandelwal,Virna Borowski,Jenny Xie,Mary Obermeier,Aberra Fura,Kevin Stefanski,Georgia Cornelius,Joseph A. Tino,John E. Macor,Luisa Salter-Cid,Rex Denton,Qihong Zhao,Percy H. Carter,T. G. Murali Dhar

ACS medicinal chemistry letters（2020）

引用26浏览0WOS引用

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作者统计

#Papers: 53

#Citation: 866

H-Index: 18

G-Index: 28

Sociability: 6

Diversity: 2

Activity: 21

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