Novel Dihydropteridinone Derivatives As Potent Inhibitors of the Understudied Human Kinases Vaccinia-Related Kinase 1 and Casein Kinase 1δ/ε
Fernando H. de Souza Gama,Luiz A. Dutra, Michael Hawgood,Caio Vinícius dos Reis,Ricardo A. M. Serafim,Marcos A. Ferreira, Bruno V. M. Teodoro,Jéssica Emi Takarada, André S. Santiago,Dimitrios-Ilias Balourdas, Ann-Sofie Nilsson, Bruno Urien, Vitor M. Almeida,Carina Gileadi, Priscila Z. Ramos, Anita Salmazo,Stanley N. S. Vasconcelos, Micael R. Cunha,Susanne Mueller,Stefan Knapp,Katlin B. Massirer, Jonathan M. Elkins,Opher Gileadi,Alessandra Mascarello, Bennie B. L. G. Lemmens, Cristiano R. W. Guimarães,Hatylas Azevedo,Rafael M. Couñago Journal of Medicinal Chemistry(2024)
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