Discovery of Icenticaftor (QBW251), a Cystic Fibrosis Transmembrane Conductance Regulator Potentiator with Clinical Efficacy in Cystic Fibrosis and Chronic Obstructive Pulmonary Disease Darren Le Grand , Martin Gosling , Urs Baettig , Parmjit Bahra , Kamlesh Bala , Cara Brocklehurst , Emma Budd , Rebecca Butler , Atwood K. Cheung , Hedaythul Choudhury , Stephen P. Collingwood , Brian Cox , Henry Danahay , Lee Edwards , Brian Everatt , Ulrike Glaenzel , Anne-Lise Glotin , Paul Groot-Kormelink , Edward Hall , Julia Hatto , Catherine Howsham , Glyn Hughes , Anna King , Julia Koehler , Swarupa Kulkarni , , Ian Nicholls , Christopher Page , Giles Pergl-Wilson , Mariana Oana Popa , Richard Robinson , David Rowlands , Tom Sharp , Matthew Spendiff , Emily Stanley , Oliver Steward , Roger J. Taylor , Pamela Tranter , Trixie Wagner , Hazel Watson , Gareth Williams , Penny Wright , Alice Young , David A. Sandham Journal of medicinal chemistry(2021)
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