Synthesis and SAR of 5-aryl-furan-2-carboxamide derivatives as potent urotensin-II receptor antagonists.
Bioorganic & Medicinal Chemistry Letters(2019)
摘要
The synthesis and SAR of 5-arylfuran-2-carboxamide derivatives as urotensin-II receptor antagonists are described.
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关键词
Urotensin-II receptor,Antagonists,5-Aryl-furan-2-carboxamide,Cardiovascular disease
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